Research Article Hua Fu Corresponding Author E-mail address: fuhua@mail.tsinghua.edu.cn Tsinghua University, Department of Chemistry, Department of Chemistry, Tsinghua University, 100084 Beijing, CHINA Search for more papers by this author PDF PDF Share Abstract Here we report a novel kind of bioorthogonal ligation and cleavage method via reactions of chloroquinoxalines (CQ) and ortho ‐dithiophenols (DT), in which double nucleophilic substitutions of ortho ‐dithiophenols to chloroquinoxalines...